LOCOID
Available from Value Pharmaceuticals at discount price
CONTRAINDICATIONS 
  
Topical corticosteroids are contraindicated in those patients with a history of hypersensitivity to any 
of the components of the preparation. 
  
PRECAUTIONS 
  
General 
  
Systemic absorption of topical corticosteroids has produced reversible 
hypothalamic-pituitary-adrenal (HPA) axis suppression, manifestations of Cushing's syndrome, 
hyperglycemia, and glucosuria in some patients. 
  
Conditions which augment systemic absorption include the application of the more potent steroids, 
use over large surface areas, prolonged use, and the addition of occlusive dressings. 
  
Therefore, patients receiving a large dose of a potent topical steroid applied to a large surface area 
or under an occlusive dressing should be evaluated periodically for evidence of HPA axis 
suppression by using the urinary free cortisol and ACTH stimulation tests. If HPA axis suppression 
is noted, an attempt should be made to withdraw the drug, to reduce the frequency of application, or 
to substitute a less potent steroid. 
  
Recovery of HPA axis function is generally prompt and complete upon discontinuation of the drug. 
Infrequently, signs and symptoms of steroid withdrawal may occur, requiring supplemental systemic 
corticosteroids. 
  
Children may absorb proportionally larger amounts of topical corticosteroids and thus be more 
susceptible to systemic toxicity. (See Pediatric Use.) If irritation develops, topical corticosteroids 
should be discontinued and appropriate therapy instituted. In the presence of dermatological 
infections, the use of an appropriate antifungal or antibacterial agent should be instituted. If a 
favorable response does not occur promptly, the corticosteroid should be discontinued until the 
infection has been adequately controlled. 
  
Information for the Patient 
  
Patients using topical corticosteroids should receive the following information and instructions: 
  
     1. This medication is to be used as directed by the physician. It is for external use only. 
     Avoid contact with the eyes. 
     2. Patients should be advised not to use this medication for any disorder other than for which 
     it was prescribed. 
     3. The treated skin area should not be bandaged or otherwise covered or wrapped as to be 
     occlusive unless directed by the physician. 
     4. Patients should report any signs of local adverse reactions especially under occlusive 
     dressing. 
     5. Parents of pediatric patients should be advised not to use tight-fitting diapers or plastic 
     pants on a child being treated in the diaper area, as these garments may constitute occlusive 
     dressings. 
  
Laboratory Tests 
  
The following tests may be helpful in evaluating the HPA axis suppression: 
  
     Urinary free cortisol test. 
     ACTH stimulation test. 
  
Carcinogenesis, Mutagenesis, and Impairment of Fertility 
  
Long-term animal studies have not been performed to evaluate the carcinogenic potential or the 
effect on fertility of topical corticosteroids. 
  
Studies to determine mutagenicity with prednisolone and hydrocortisone have revealed negative 
results. 
  
Pregnancy Category C 
  
Corticosteroids are generally teratogenic in laboratory animals when administered systemically at 
relatively low dosage levels. The more potent corticosteroids have been shown to be teratogenic 
after dermal application in laboratory animals. There are no adequate and well-controlled studies in 
pregnant women on teratogenic effects from topically applied corticosteroids. Therefore, topical 
corticosteroids should be used during pregnancy only if the potential benefit justifies the potential 
risk to the fetus. Drugs of this class should not be used extensively on pregnant patients, in large 
amounts, or for prolonged periods of time. 
  
Nursing Mothers 
  
It is not known whether topical administration of corticosteroids could result in sufficient systemic 
absorption to produce detectable quantities in breast milk. Systemically administered corticosteroids 
are secreted into breast milk in quantities not likely to have a deleterious effect on the infant. 
Nevertheless, caution should be exercised when topical corticosteroids are administered to a nursing 
woman. 
  
Pediatric Use 
  
Pediatric patients may demonstrate greater susceptibility to topical corticosteroid-induced 
HPA axis suppression and Cushing's syndrome than mature patients because of a larger skin 
surface area to body weight ratio. 
  
Hypothalamic-pituitary-adrenal (HPA) axis suppression, Cushing's syndrome, and intracranial 
hypertension have been reported in children receiving topical corticosteroids. 
  
Manifestations of adrenal suppression in children include linear growth retardation, delayed weight 
gain, low plasma cortisol levels, and absence of response to ACTH stimulation. Manifestations of 
intracranial hypertension include bulging fontanelles, headaches, and bilateral papilledema. 
  
Administration of topical corticosteroids to children should be limited to the least amount compatible 
with an effective therapeutic regimen. Chronic corticosteroid therapy may interfere with the growth 
and development of children.